Pharm
Gonadotropin-releasing Hormone Agonist
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Gonadotropin-releasing Hormone Agonist
, GnRH agonist, Nafarelin Acetate, Synarel
Indication
Endometriosis
Pathophysiology
Potentiates Gonadotropin-releasing
Hormone
(GnRH)
Results in hypoestrogenism or pseudo-
Menopause
Does not cause the same androgenic effects as
Danazol
Dosing
Nafarelin Acetate (Synarel)
Synarel 200-400 micro-g intranasally bid
Efficacy
Effective at regression of lesions and relief of pain
No proven effect on fertility
Adverse effects
Menopausal symptoms
Hot Flashes
Insomnia
Emotional changes
Bone density loss with prolonged use
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