• Physiology
  1. Transport Proteins aid in substance transfer in and out of the cell
  • Pathophysiology
  1. Transport Proteins may interfere with drug absorption, distribution and elimination
  • Types
  1. Breast Cancer Resistance Protein (BCRP)
  2. Organic Anion Transport Protein (e.g. OATP1B1, OATP1B3)
  3. Organic Cation Transport Protein (e.g. OCT2)
  4. Multidrug and Toxin Exctrusion Protein (e.g. MATE1, MAE2-K)
  • References
  1. (2022) presc lett 29(8): 47-8